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Publication --> 2018

"Exploiting ]Amino Acid Enolates in Direct Catalytic Diastereo] and Enantioselective C]C Bond Forming Reactions"
Yu, J.-S.; Noda, H.; Shibasaki, M.
Chem. Eur. J. 2018, 24, 15796.


"anti-Selective Catalytic Asymmetric Nitroaldol Reaction of -Keto Esters; Intriguing Solvent Effect, Flow Reaction, and Synthesis of APIs"
Karasawa, T.; Oriez, R.; Kumagai, N.; Shibasaki, M.
J. Am. Chem. Soc. 2018, 140, 12290.


"Structure-activity relationship study of leucinostatin A, a modulator of tumor|stroma interaction"
Abe, H.; Kawada, M.; Sakashita, C.; Watanabe, T.; Shibasaki, M.
Tetrahedron 2018, 74, 5129.


"Direct Catalytic Asymmetric 1,6-Conjugate Addition of Amides to p-Quinone Methides"
Sun, Z.; Sun, B.; Kumagai, N.; Shibasaki, M.
Org. Lett. 2018, 20, 3070.


"Direct Catalytic Asymmetric Aldol Reaction of -Vinyl Acetamide"
Takeuchi, T.; Kumagai, N.; Shibasaki, M.
J. Org. Chem. 2018, 83, 5851.


"Direct enolization chemistry of 7-azaindoline amides: A case study of bis(tetrahydrophosphole)-type ligands"
Li, Z.; Noda, H.; Kumagai, N.; Shibasaki, M.
Tetrahedron 2018, 74, 3301.


"Catalytic Asymmetric Synthesis of -Trifluoromethylated Carbinols: A Case Study of Tertiary Propargylic Alcohols"
Noda, H.; Kumagai, N.; Shibasaki, M.
Asian J. Org. Chem. 2018, 7, 599.


"Conquering amide planarity: structural distortion and its hidden reactivity"
Adachi, S.; Kumagai, N.; Shibasaki, M.
Tetrahedron Lett. 2018, 59, 1147.


"Catalytic Oligopeptide Synthesis"
Liu, Z.; Noda, H.; Shibasaki, M.; Kumagai, N.
Org. Lett. 2018, 20, 612.


"Direct Catalytic Asymmetric Mannich-Type Reaction en Route to -Hydroxy--amino Acid Derivatives"
Sun, B.; Pluta, R.; Kumagai, N.; Shibasaki, M.
Org. Lett. 2018, 20, 526.


"Direct Catalytic Asymmetric Aldol Reaction of Thioamide with an -Vinyl Appendage"
Cui, J.; Ohtsuki, A.; Watanabe, T.; Kumagai, N.; Shibasaki, M.
Chem. Eur. J. 2018, 24, 2598.


"Heterogeneous Heterobimetallic Catalysis Enabling Expeditious Access to CF3-Containing vic-Amino Alcohols"
Karasawa, T.; Kumagai, N.; Shibasaki, M.
Org. Lett. 2018, 20, 308.


"Quaternary 2,2-Amino Acids: Catalytic Asymmetric Synthesis and Incorporation into Peptides by Fmoc-Based Solid-Phase Peptide Synthesis"
Yu, J.-S.; Noda, H.; Shibasaki, M.
Angew. Chem. Int. Ed. 2018, 57, 818.


Synthetic studies of viridiofungins, broad-spectrum antifungal agents and serine palmitoyl transferase inhibitors
Kumagai, N.; Shibasaki, M.
J. Antibiot. 2018, 71, 53.



"Structural and Computational Investigation of Intramolecular N...H Interactions in - and -Fluorinated 7-Azaindoline Amides"
Brewitz, L.; Noda, H.; Kumagai, N.; Shibasaki, M.
Eur. J. Org. Chem. 2018, 714. Selected as a front cover.


"Bis(2-pyridyl)amides as Readily Cleavable Amides Under Catalytic, Neutral, and Room-Temperature Conditions"
Adachi, S.; Kumagai, N.; Shibasaki, M.
Synlett 2018, 29, 301.